High affinity apelin receptor agonist. Binds apelin receptors in left ventricle from normal and pulmonary arterial hypertensive (PAH) hearts (pKi values are 9.31 and 9.46, respectively). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro.

硫辛酰胺是 6,8-二硫代辛酰胺的俗名。

Calpain Inhibitor III 是一种有效的细胞渗透性钙蛋白酶 I 和 II 抑制剂 (Ki = 8 nM)。Calpain Inhibitor III（也参考 CAS 88191-84-8）可控制钙蛋白酶的生物活性。